ActiTide™ AH3 / Acetyl Hexapeptide-8

Kufotokozera Kwachidule:

ActiTide™ AH3 ndi chidutswa cha hexapeptide chomwe chimatsanzira kapangidwe ka puloteni ya SNAP-25. Chimapikisana ndi SNAP-25, kuletsa kupangika kwa SNARE complex ndi syntaxin ndi VAMP. Kutseka kumeneku kumaletsa kusakanikirana kwa membrane ndi kutulutsidwa kwa ma neurotransmitters. Monga chophatikizira chochepetsa makwinya mwachangu, ActiTide™ AH3 imachepetsa makwinya amphamvu omwe amayamba chifukwa cha kupindika kwa minofu ndipo imathandizira kuchepetsa kuchuluka ndi kuzama kwa mizere yowonetsera. Kuphatikiza apo, ndi yofatsa, yopanda poizoni, ndipo yoyenera mitundu yonse ya khungu. ActiTide™ AH3 imagwiritsidwa ntchito kwambiri pazinthu zokongoletsera ndi zosamalira khungu, kuphatikiza ma seramu oletsa makwinya, mafuta odzola nkhope, mafuta odzola maso, zodzoladzola zoyambira, ndi zophimba nkhope, zomwe zimapereka zabwino zonse zotsutsana ndi ukalamba.


Tsatanetsatane wa Zamalonda

Ma tag a Zamalonda

Dzina la kampani ActiTide™ AH3
Nambala ya CAS 616204-22-9
Dzina la INCI Acetyl Hexapeptide-8
Kugwiritsa ntchito Lotion, Serum, Chigoba, Chotsukira nkhope
Phukusi 100g/botolo, 1kg/thumba
Maonekedwe Ufa woyera mpaka woyera pang'ono
Kusungunuka Madzi osungunuka
Ntchito Mndandanda wa Peptide
Nthawi yosungira zinthu zaka 2
Malo Osungirako Sungani chidebecho motsekedwa bwino pamalo ozizira komanso ouma pa 2 - 8°C.
Mlingo 0.005-0.05%

Kugwiritsa ntchito

 

Kafukufuku wokhudza njira zoyambira zotsutsana ndi makwinya adapangitsa kuti ActiTide™ AH3, hexapeptide yatsopano yomwe idapangidwa kudzera mu njira yasayansi kuyambira pakupanga mwanzeru mpaka kupanga GMP, ndi zotsatira zabwino.

ActiTide™ AH3 imapereka mphamvu yochepetsera makwinya mofanana ndi Botulinum Toxin Type A, pomwe imapewa zoopsa za jakisoni ndikupereka ndalama zambiri.

 

Ubwino Wokongoletsa:

ActiTide™ AH3 imachepetsa kuzama kwa makwinya komwe kumachitika chifukwa cha kupindika kwa minofu ya nkhope, zomwe zimakhudza kwambiri pamphumi ndi m'mitsempha ya m'mimba.

 

Njira Yogwirira Ntchito:

Kupindika kwa minofu kumachitika pamene neurotransmitter yatulutsidwa kuchokera ku synaptic vesicles. SNARE complex - gulu la mapuloteni a VAMP, Syntaxin, ndi SNAP-25 - ndi lofunikira kwambiri pakupanga vesicle docking ndi neurotransmitter exocytosis (A. Ferrer Montiel et al., JBC 1997, 272:2634-2638). Complex iyi imagwira ntchito ngati mbedza ya ma cell, kugwira ma vesicles ndikuyendetsa membrane fusion.

Monga chitsanzo cha kapangidwe ka SNAP-25 N-terminus, ActiTide™ AH3 imapikisana ndi SNAP-25 kuti ilowe mu SNARE complex, zomwe zimapangitsa kuti igwirizane. Kusokonekera kwa SNARE complex kumasokoneza kutsekeka kwa vesicle ndi kutulutsidwa kwa neurotransmitter pambuyo pake, zomwe zimapangitsa kuti minofu ichepetse komanso kupewa makwinya ndi mapangidwe a mizere yaying'ono.

ActiTide™ AH3 ndi njira yotetezeka, yotsika mtengo, komanso yofewa m'malo mwa Botulinum Toxin Type A. Imalimbana ndi njira yomweyo yopangira makwinya koma imagwira ntchito mwanjira yosiyana.


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