ActiTide-AH3 / Acetyl Hexapeptide-8

Kufotokozera Kwachidule:

ActiTide-AH3 ndi chidutswa cha hexapeptide chomwe chimatengera kapangidwe ka mapuloteni a SNAP-25. Imapikisana ndi SNAP-25, kuletsa mapangidwe a SNARE complex ndi syntaxin ndi VAMP. Kutsekeka kumeneku kumalepheretsa kuphatikizika kwa nembanemba komanso kutulutsidwa kotsatira kwa ma neurotransmitters. Monga chinthu chochepetsera makwinya nthawi yomweyo, ActiTide-AH3 imachepetsa bwino makwinya osinthika omwe amayamba chifukwa cha kukangana kwa minofu komwe amakhala ndipo amathandizira kuchepetsa kuchuluka ndi kuya kwa mizere yofotokozera. Kuphatikiza apo, ndi yofatsa, yopanda poizoni, komanso yoyenera pakhungu lamitundu yonse. ActiTide-AH3 imagwiritsidwa ntchito kwambiri pazinthu zodzikongoletsera komanso zosamalira khungu, kuphatikiza ma seramu oletsa makwinya, mafuta opaka kumaso, zopaka m'maso, zodzoladzola zoyambira, ndi masks, zomwe zimapereka zabwino zambiri zoletsa kukalamba.


Tsatanetsatane wa Zamalonda

Zolemba Zamalonda

Dzina lamalonda ActiTide-AH3
CAS No. 616204-22-9
Dzina la INCI Acetyl Hexapeptide-8
Kugwiritsa ntchito Mafuta odzola, seramu, chigoba, zotsukira nkhope
Phukusi 100g / botolo, 1kg / thumba
Maonekedwe Ufa woyera mpaka woyera
Kusungunuka Madzi sungunuka
Ntchito Peptide mndandanda
Alumali moyo zaka 2
Kusungirako Sungani chidebecho chotsekedwa mwamphamvu m'malo ozizira, owuma pa 2 - 8 ° C.
Mlingo 0.005-0.05%

Kugwiritsa ntchito

Kafukufuku wokhudzana ndi njira zolimbana ndi makwinya adapangitsa kuti atulutsidwe ActiTide-AH3, hexapeptide yopangidwa mwaluso kudzera munjira yasayansi kuchokera ku kapangidwe koyenera mpaka kupanga GMP, ndi zotsatira zabwino.

ActiTide-AH3 imapereka mphamvu yochepetsera makwinya yofanana ndi Mtundu A wa Toxin wa Botulinum, kwinaku ikupewa kuopsa kwa jakisoni komanso kupereka ndalama zochulukirapo.

Ubwino Wodzikongoletsa:
ActiTide-AH3 imachepetsa kuya kwa makwinya komwe kumachitika chifukwa cha kukangana kwa minofu ya nkhope, zomwe zimawonekera pamphumi ndi makwinya a periocular.

Kachitidwe Kachitidwe:
Kudumpha kwa minofu kumachitika pakatulutsidwa kwa ma neurotransmitter kuchokera ku ma synaptic vesicles. The SNARE complex - msonkhano wa ternary wa VAMP, Syntaxin, ndi SNAP-25 mapuloteni - ndizofunikira pa vesicle docking ndi neurotransmitter exocytosis (A. Ferrer Montiel et al., JBC 1997, 272: 2634-2638). Zovutazi zimakhala ngati mbedza yama cell, kugwira ma vesicles ndikuyendetsa kaphatikizidwe ka membrane.

Monga chojambula chojambula cha SNAP-25 N-terminus, ActiTide-AH3 imapikisana ndi SNAP-25 kuti iphatikizidwe mu zovuta za SNARE, ndikuwongolera msonkhano wake. Kuwonongeka kwa zovuta za SNARE kumapangitsa kuti vesicle docking iwonongeke komanso kutulutsidwa kwa ma neurotransmitter, zomwe zimapangitsa kuchepa kwa minofu ndikupewa makwinya ndi kupanga mizere yabwino.

ActiTide-AH3 ndi njira yotetezeka, yotsika mtengo, komanso yochepetsetsa kusiyana ndi Botulinum Toxin Type A. Imayang'ana njira yomweyo yopangira makwinya koma imagwira ntchito mosiyanasiyana.


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