Dzina lamalonda | ActiTide™ AH3 |
CAS No. | 616204-22-9 |
Dzina la INCI | Acetyl Hexapeptide-8 |
Kugwiritsa ntchito | Mafuta odzola, ma seramu, masks, oyeretsa nkhope |
Phukusi | 100g / botolo, 1kg / thumba |
Maonekedwe | Ufa woyera mpaka woyera |
Kusungunuka | Madzi sungunuka |
Ntchito | Peptide mndandanda |
Alumali moyo | zaka 2 |
Kusungirako | Sungani chidebecho chotsekedwa mwamphamvu pamalo ozizira, owuma pa 2 - 8 ° C. |
Mlingo | 0.005-0.05% |
Kugwiritsa ntchito
Kafukufuku wokhudzana ndi njira zothana ndi makwinya adapangitsa kuti ActiTide™ AH3, hexapeptide yopangidwa mwanzeru yopangidwa kudzera munjira yasayansi kuchokera pakupanga koyenera mpaka kupanga GMP, ndi zotsatira zabwino.
ActiTide™ AH3 imapereka mphamvu yochepetsera makwinya yofanana ndi Botulinum Toxin Type A, kwinaku ikupewa kuopsa kwa jakisoni komanso kupereka ndalama zambiri.
Ubwino Wodzikongoletsa:
ActiTide™ AH3 imachepetsa kuya kwa makwinya komwe kumachitika chifukwa cha kukangana kwa minofu ya nkhope, ndi zotsatira zowonekera pamphumi ndi makwinya a periocular.
Njira Yochitira:
Kutsika kwa minofu kumachitika pamene neurotransmitter imatulutsidwa kuchokera ku ma synaptic vesicles. The SNARE complex - msonkhano wa ternary wa VAMP, Syntaxin, ndi SNAP-25 mapuloteni - ndizofunikira pa vesicle docking ndi neurotransmitter exocytosis (A. Ferrer Montiel et al., JBC 1997, 272: 2634-2638). Zovutazi zimakhala ngati mbedza yama cell, kugwira ma vesicles ndikuyendetsa kaphatikizidwe ka membrane.
Monga chojambula chojambula cha SNAP-25 N-terminus, ActiTide™ AH3 imapikisana ndi SNAP-25 kuti iphatikizidwe mu zovuta za SNARE, ndikuwongolera msonkhano wake. Kuwonongeka kwa zovuta za SNARE kumapangitsa kuti vesicle docking iwonongeke komanso kutulutsidwa kwa ma neurotransmitter, zomwe zimapangitsa kuchepa kwa minofu ndikupewa makwinya ndi kupanga mizere yabwino.
ActiTide™ AH3 ndi njira yotetezeka, yotsika mtengo, komanso yofatsa kuposa ya Botulinum Toxin Type A. Imalunjika panjira yomweyi yopangira makwinya koma imagwira ntchito mosiyanasiyana.