ActiTide™ AH3 / Acetyl Hexapeptide-8

Kufotokozera Kwachidule:

ActiTide™ AH3 ndi chidutswa cha hexapeptide chomwe chimatengera kapangidwe ka mapuloteni a SNAP-25. Imapikisana ndi SNAP-25, kuletsa mapangidwe a SNARE complex ndi syntaxin ndi VAMP. Kutsekeka kumeneku kumalepheretsa kuphatikizika kwa nembanemba komanso kutulutsidwa kotsatira kwa ma neurotransmitters. Monga chopangira chochepetsera makwinya pompopompo, ActiTide™ AH3 imachepetsa bwino makwinya omwe amayamba chifukwa cha kugundana kwa minofu komwe amakhala ndikuthandizira kuchepetsa kuchuluka ndi kuya kwa mizere yofotokozera. Kuphatikiza apo, ndi yofatsa, yopanda poizoni, komanso yoyenera pakhungu lamitundu yonse. ActiTide™ AH3 imagwiritsidwa ntchito kwambiri pazokongoletsa komanso zosamalira khungu, kuphatikiza ma seramu oletsa makwinya, zopaka kumaso, zopaka m'maso, zopakapaka pansi, ndi masks, zomwe zimapereka zabwino zambiri zoletsa kukalamba.


Tsatanetsatane wa Zamalonda

Zolemba Zamalonda

Dzina lamalonda ActiTide™ AH3
CAS No. 616204-22-9
Dzina la INCI Acetyl Hexapeptide-8
Kugwiritsa ntchito Mafuta odzola, ma seramu, masks, oyeretsa nkhope
Phukusi 100g / botolo, 1kg / thumba
Maonekedwe Ufa woyera mpaka woyera
Kusungunuka Madzi sungunuka
Ntchito Peptide mndandanda
Alumali moyo zaka 2
Kusungirako Sungani chidebecho chotsekedwa mwamphamvu pamalo ozizira, owuma pa 2 - 8 ° C.
Mlingo 0.005-0.05%

Kugwiritsa ntchito

 

Kafukufuku wokhudzana ndi njira zothana ndi makwinya adapangitsa kuti ActiTide™ AH3, hexapeptide yopangidwa mwanzeru yopangidwa kudzera munjira yasayansi kuchokera pakupanga koyenera mpaka kupanga GMP, ndi zotsatira zabwino.

ActiTide™ AH3 imapereka mphamvu yochepetsera makwinya yofanana ndi Botulinum Toxin Type A, kwinaku ikupewa kuopsa kwa jakisoni komanso kupereka ndalama zambiri.

 

Ubwino Wodzikongoletsa:

ActiTide™ AH3 imachepetsa kuya kwa makwinya komwe kumachitika chifukwa cha kukangana kwa minofu ya nkhope, ndi zotsatira zowonekera pamphumi ndi makwinya a periocular.

 

Njira Yochitira:

Kutsika kwa minofu kumachitika pamene neurotransmitter imatulutsidwa kuchokera ku ma synaptic vesicles. The SNARE complex - msonkhano wa ternary wa VAMP, Syntaxin, ndi SNAP-25 mapuloteni - ndizofunikira pa vesicle docking ndi neurotransmitter exocytosis (A. Ferrer Montiel et al., JBC 1997, 272: 2634-2638). Zovutazi zimakhala ngati mbedza yama cell, kugwira ma vesicles ndikuyendetsa kaphatikizidwe ka membrane.

Monga chojambula chojambula cha SNAP-25 N-terminus, ActiTide™ AH3 imapikisana ndi SNAP-25 kuti iphatikizidwe mu zovuta za SNARE, ndikuwongolera msonkhano wake. Kuwonongeka kwa zovuta za SNARE kumapangitsa kuti vesicle docking iwonongeke komanso kutulutsidwa kwa ma neurotransmitter, zomwe zimapangitsa kuchepa kwa minofu ndikupewa makwinya ndi kupanga mizere yabwino.

ActiTide™ AH3 ndi njira yotetezeka, yotsika mtengo, komanso yofatsa kuposa ya Botulinum Toxin Type A. Imalunjika panjira yomweyi yopangira makwinya koma imagwira ntchito mosiyanasiyana.


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