ActiTide-PT7 / Palmitoyl Tetrapeptide-7

Kufotokozera Kwachidule:

Immunoglobulin G (IgG) ndiye gawo lalikulu la ma immunoglobulins mu seramu yamunthu komanso antibody yochuluka kwambiri m'thupi. ActiTide-PT7 ndi chochokera palmitoylated cha Gly-Gln-Pro-Arg (GQPR) tetrapeptide, yochokera ku chidutswa (341-344) cha immunoglobulin G heavy chain. Kafukufuku wasonyeza kuti GQPR tetrapeptide imatha kulimbikitsa macrophages ndi neutrophils, kupititsa patsogolo ntchito ya phagocytic. Kuphatikiza apo, GQP ndi njira yodziwika bwino ya tripeptide yomwe imapezeka mumtundu wa IV collagen. Monga wothandizira khungu, ActiTide-PT7 ikhoza kulepheretsa kutulutsa kwa cytokines (IL-6), kulimbikitsa kaphatikizidwe ka laminin, fibronectin, ndi collagen, kuchepetsa makwinya a khungu, ndipo kumakhala ndi zotsatira zotsitsimula komanso zolimbikitsa.


Tsatanetsatane wa Zamalonda

Zolemba Zamalonda

Dzina lamalonda ActiTide-PT7
CAS No. 221227-05-0
Dzina la INCI Palmitoyl Tetrapeptide-7
Kugwiritsa ntchito Mafuta odzola, seramu, chigoba, zotsukira nkhope
Phukusi 100g / botolo
Maonekedwe Ufa woyera mpaka woyera
Kusungunuka Zosasungunuka m'madzi
Ntchito Peptide mndandanda
Alumali moyo zaka 2
Kusungirako Sungani chidebecho chotsekedwa mwamphamvu m'malo ozizira, owuma pa 2 - 8 ° C.
Mlingo 0.001-0.1% pansi pa 45 °C

Kugwiritsa ntchito

ActiTide-PT7 ndi peptide yogwira ntchito yomwe imatsanzira chidutswa cha immunoglobulin IgG. Kusinthidwa ndi palmitoylation, imawonetsa kukhazikika kokhazikika komanso mphamvu ya mayamwidwe a transdermal, zomwe zimapangitsa kulowa bwino pakhungu kuti lichite ntchito yake.

Core Mechanism of Action: Kuwongolera Kutupa:

Kuwongolera Chinthu Chofunika Kwambiri: Njira yake yaikulu imakhala yochepetsera kwambiri kupanga cytokine Interleukin-6 (IL-6).

Kuchepetsa Kuyankha Kwachifuwa: IL-6 ndi mkhalapakati wofunikira pamayendedwe otupa pakhungu. Kuchuluka kwa IL-6 kumakulitsa kutupa, kumathandizira kuwonongeka kwa collagen ndi mapuloteni ena ofunikira pakhungu, potero amalimbikitsa ukalamba wa khungu. Palmitoyl Tetrapeptide-7 imagwira ntchito pakhungu la keratinocyte ndi ma fibroblasts kudzera pakukondoweza kwazizindikiro, kuwongolera mayankho otupa, makamaka poletsa kutulutsa kwambiri kwa IL-6 ku maselo oyera amagazi.

Dose-Dependent Inhibition: Maphunziro a labotale amatsimikizira kuti amalepheretsa kupanga IL-6 modalira mlingo; Kuchulukirachulukira kumabweretsa zolepheretsa kwambiri (mpaka 40% kuchuluka kwa zoletsa).

Zothandiza Kwambiri Polimbana ndi Kuwonongeka kwa Zithunzi: Nthawi yomwe ma radiation ya ultraviolet (UV) imapangitsa kupanga kwakukulu kwa IL-6, maselo omwe amathandizidwa ndi Palmitoyl Tetrapeptide-7 amawonetsa kuletsa kwa IL-6 kupanga mpaka 86%.

Zothandiza Kwambiri ndi Zopindulitsa:

Amatsitsimutsa ndi Kuchepetsa Kutupa: Poletsa mogwira mtima zinthu zotupa monga IL-6, zimachepetsa zotupa zosayenera zapakhungu, kuchepetsa kufiira komanso kusapeza bwino.

Imateteza Ku Kuwonongeka Kwa Chilengedwe: Imathandiza kuti ma cytokines asamayende bwino, kuteteza khungu ku kuwonongeka kwa chilengedwe (monga ma radiation a UV) ndi kuwonongeka kwa glycation.

Imalimbikitsa Ngakhale Khungu Lalikulu: Kuchepetsa kutupa kumathandiza kuti khungu likhale lofiira komanso zovuta zina zosagwirizana, zomwe zimathandiza kuti khungu likhale lowala kwambiri.

Kuchedwa Zizindikiro za Ukalamba: Pochepetsa kutupa ndikuletsa kuwonongeka kwa collagen, zimathandiza kuthana ndi zizindikiro za ukalamba monga makwinya ndi kugwa.

Synergistic Enhancement: Ikaphatikizidwa ndi zinthu zina zogwira ntchito (monga Palmitoyl Tripeptide-1), mwachitsanzo mu Matrixyl 3000 complex, imapanga synergistic zotsatira, kupititsa patsogolo zotsatira zotsutsa kukalamba.

Ntchito:

ActiTide-PT7 imagwiritsidwa ntchito kwambiri pazinthu zosamalira khungu, makamaka imagwira ntchito yofunika kwambiri pakukonza khungu, zoziziritsa kukhosi, komanso zolimbitsa thupi.


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